AMG-076 structure
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Common Name | AMG-076 | ||
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CAS Number | 693823-79-9 | Molecular Weight | 462.54800 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C26H33F3N2O2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of AMG-076AMG-076 is a potent, selective, non-peptide antagonist of MCHR1 (Melanin-concentrating hormone receptor 1) with binding IC50 of 0.6 nM, with dramatically reduced hERG liability (IC50>5 uM). |
Name | 1-[2-[(4aR,11R,11aS)-11-methyl-9-(trifluoromethyl)-1,3,4,4a,5,6,11,11a-octahydropyrido[4,3-b]carbazol-2-yl]ethyl]cyclohexane-1-carboxylic acid |
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Synonym | More Synonyms |
Molecular Formula | C26H33F3N2O2 |
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Molecular Weight | 462.54800 |
Exact Mass | 462.24900 |
PSA | 56.33000 |
LogP | 6.14750 |
UNII-HX4T7JEV3D |
AMG-076 free base |
AMG 076 |