PKC-IN-7 structure
|
Common Name | PKC-IN-7 | ||
---|---|---|---|---|
CAS Number | 860468-10-6 | Molecular Weight | 443.931 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C26H22ClN3O2 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of PKC-IN-7PKC-IN-7 is a potent, selective, reversible, ATP-competitive PKCα/β inhibitor with IC50 of 4.7/3.3 nM; dispalys >50-fold selectivity against PKC isotypes δ,ε,η,θ and other kinases belonging to the AGC family; inhibits IgM-stimulated mouse B cell proliferation with an IC50 of 296 nM. |
Name | PKC-IN-7 |
---|
Description | PKC-IN-7 is a potent, selective, reversible, ATP-competitive PKCα/β inhibitor with IC50 of 4.7/3.3 nM; dispalys >50-fold selectivity against PKC isotypes δ,ε,η,θ and other kinases belonging to the AGC family; inhibits IgM-stimulated mouse B cell proliferation with an IC50 of 296 nM. |
---|---|
References | References 1. van Eis MJ, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):781-786. View Related Products by Target PKC |
Molecular Formula | C26H22ClN3O2 |
---|---|
Molecular Weight | 443.931 |