![]() PKM2 activator 3 structure
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Common Name | PKM2 activator 3 | ||
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CAS Number | 1346113-84-5 | Molecular Weight | 372.77 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C15H11ClF2N2O3S | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of PKM2 activator 3PKM2 activator 3 is a potent PKM2 activator with an AC50 value of 90 nM. PKM2 activator 3 has good Caco-2 permeability, a low efflux ratio and high microsomal stability. PKM2 activator 3 can be used for researching anticancer[1]. (AC50: the concentration which gives 50% activation of enzyme.) |
Name | PKM2 activator 3 |
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Description | PKM2 activator 3 is a potent PKM2 activator with an AC50 value of 90 nM. PKM2 activator 3 has good Caco-2 permeability, a low efflux ratio and high microsomal stability. PKM2 activator 3 can be used for researching anticancer[1]. (AC50: the concentration which gives 50% activation of enzyme.) |
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Related Catalog | |
Target |
PKM2[1] |
In Vivo | PKM2 activator 3 (compound 66) has good Caco-2 permeability, a low efflux ratio (0.84) and high microsomal stability (t1/2 = 277.2 min in human liver microsomes and 117.5 min in mouse liver microsomes)[1]. |
References |
Molecular Formula | C15H11ClF2N2O3S |
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Molecular Weight | 372.77 |