BPTF-IN-1

Modify Date: 2024-01-09 18:37:09

BPTF-IN-1 Structure
BPTF-IN-1 structure
Common Name BPTF-IN-1
CAS Number 2359618-49-6 Molecular Weight 450.47
Density N/A Boiling Point N/A
Molecular Formula C23H23FN6O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of BPTF-IN-1


BPTF-IN-1 (compound AU1) is a selective bromodomain and PHD finger containing transcription factor (BPTF) bromodomain inhibitor with a Kd of 2.8 μM. BPTF-IN-1 shows to be selective for BPTF over BRD4 bromodomain. BPTF-IN-1 shows antimalarial activity[1].

 Names

Name BPTF-IN-1

 BPTF-IN-1 Biological Activity

Description BPTF-IN-1 (compound AU1) is a selective bromodomain and PHD finger containing transcription factor (BPTF) bromodomain inhibitor with a Kd of 2.8 μM. BPTF-IN-1 shows to be selective for BPTF over BRD4 bromodomain. BPTF-IN-1 shows antimalarial activity[1].
Related Catalog
References

[1]. Steven E Kirberger, et al. Selectivity, ligand deconstruction, and cellular activity analysis of a BPTF bromodomain inhibitor. Org Biomol Chem. 2019 Feb 13;17(7):2020-2027.

 Chemical & Physical Properties

Molecular Formula C23H23FN6O3
Molecular Weight 450.47