ALK5-IN-27 structure
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Common Name | ALK5-IN-27 | ||
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CAS Number | 2785430-83-1 | Molecular Weight | 440.54 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C25H28N8 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of ALK5-IN-27ALK5-IN-27 (Compound EX-04) is a potent ALK-5 inhibitor with an IC50 ≤10 nM. ALK5-IN-27 also inhibits ALK-2 (selectivity ALK2/ALK5 ≤10)[1]. |
Name | ALK5-IN-27 |
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Description | ALK5-IN-27 (Compound EX-04) is a potent ALK-5 inhibitor with an IC50 ≤10 nM. ALK5-IN-27 also inhibits ALK-2 (selectivity ALK2/ALK5 ≤10)[1]. |
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Related Catalog | |
Target |
ALK5:≤10 nM (IC50) ALK2 |
References |
[1]. Bettina FRANZ, et al. Alk-5 inhibitors and uses thereof. Patent WO2022126133A1. |
Molecular Formula | C25H28N8 |
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Molecular Weight | 440.54 |