1175273-62-7

• 常用中文名：1-(4-哌啶基)-1H-吡唑-4-硼酸频那醇盐酸盐
• 常用英文名：4-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]piperidine,hydrochloride
• CAS号：1175273-62-7
• 分子式：C₁₄H₂₅BClN₃O₂
• 分子量：313.63100
• 发布时间：2018-10-21 17:03:08
• 更新时间：2024-06-21 17:50:06

名称

• 中文名: 1-(4-哌啶基)-1H-吡唑-4-硼酸频那醇盐酸盐
• 英文名: 4-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]piperidine,hydrochloride

物化性质

• 分子式: C₁₄H₂₅BClN₃O₂
• 分子量: 313.63100
• 精确质量: 313.17300
• PSA: 48.31000
• LogP: 2.23760

合成路线

877399-74-1 ~99% 1175273-62-7

文献：OSI PHARMACEUTICALS, LLC; HOMBERGER, Keith, R.; BERGER, Dan, M.; CHEN, Xin; CREW, Andrew, P.; DONG, Hanqing; KLEINBERG, Andrew; LI, An-Hu; MA, Lifu; MULVIHILL, Mark, J.; PANICKER, Bijoy; SIU, Kam, W.; STEINIG, Arno, G.; TARRANT, James, G.; WANG, Jing; WENG, Qinghua; SANGEM, Rajaram; GUPTA, Ramesh, C. Patent: WO2011/100502 A1, 2011 ; Location in patent: Page/Page column 42 ; WO 2011/100502 A1

109384-19-2 ~% 1175273-62-7

文献：HUTCHISON MEDIPHARMA LIMITED; Su, Wei-Guo; Deng, Wei; Ji, Jianguo Patent: US2014/121200 A1, 2014 ;

141699-59-4 ~% 1175273-62-7

文献：HUTCHISON MEDIPHARMA LIMITED; Su, Wei-Guo; Deng, Wei; Ji, Jianguo Patent: US2014/121200 A1, 2014 ;

269410-08-4 ~% 1175273-62-7

文献：OSI PHARMACEUTICALS, LLC; LI, An-Hu; MULVIHILL, Mark, J.; STEINIG, Arno, G. Patent: WO2011/143646 A1, 2011 ; WO 2011/143646 A1