Bromodomain inhibitor-10

Modify Date: 2024-01-23 14:00:09

Bromodomain inhibitor-10 Structure
Bromodomain inhibitor-10 structure
Common Name Bromodomain inhibitor-10
CAS Number 1870849-58-3 Molecular Weight 364.40
Density N/A Boiling Point N/A
Molecular Formula C20H20N4O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Bromodomain inhibitor-10


Bromodomain inhibitor-10 (compound 128) is a potent bromodomain inhibitor with Kds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40[1].

 Names

Name Bromodomain inhibitor-10

 Bromodomain inhibitor-10 Biological Activity

Description Bromodomain inhibitor-10 (compound 128) is a potent bromodomain inhibitor with Kds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40[1].
Related Catalog
Target

BRD4-1:15 nM (Kd)

BRD4-2:2500 nM (Kd)

References

[1]. Jimmi GERNER SEITZBERG, et al. Compounds active towards bromodomains. WO2016016316A1

 Chemical & Physical Properties

Molecular Formula C20H20N4O3
Molecular Weight 364.40