MAPK13-IN-1

Names

[ CAS No. ]:
229002-10-2

[ Name ]:
MAPK13-IN-1

Biological Activity

[Description]:

MPAK13-IN-1 is a MAPK13 (p38δ) inhibitor, with an IC50 of 620 nM.

[Related Catalog]:

Signaling Pathways >> MAPK/ERK Pathway >> p38 MAPK

Research Areas >> Others

[Target]

MAPK13 (p38δ):620 nM (IC50)

[References]

[1]. Yurtsever Z, et al. First comprehensive structural and biophysical analysis of MAPK13 inhibitors targeting DFG-in and DFG-out binding modes. Biochim Biophys Acta. 2016 Nov;1860(11 Pt A):2335-2344.

[Related Small Molecules]

SB203580 | SB202190 (FHPI) | Doramapimod (BIRB 796) | LY2228820 | SB 239063 | Losmapimod | PD 169316 | Talmapimod | Tat-NR2B9c | Dehydrocorydaline chloride | TAK-715 | VX 702 | VX-745 | SKF 86002 | Acumapimod

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₀H₂₃N₅O₂

[ Molecular Weight ]:
365.43

MAPK13-IN-1

Names

Biological Activity

Chemical & Physical Properties

Related Compounds