N-0861 racemate

Names

[ CAS No. ]:
121241-87-0

[ Name ]:
N-0861 racemate

[Synonym ]:
9H-Purin-6-amine, N-bicyclo[2.2.1]hept-2-yl-9-methyl-
N-(Bicyclo[2.2.1]hept-2-yl)-9-methyl-9H-purin-6-amine
9H-Purin-6-amine, N-bicyclo(2.2.1)hept-2-yl-9-methyl-, endo-(±)-

Biological Activity

[Description]:

N-0861 racemate is the racemate of N-0861. N-0861 is a selective adenosine A1 receptor antagonist.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Adenosine Receptor
Research Areas >> Others

[Target]

Adenosine receptor[1][2]


[References]

[1]. D.T.Witte, et al. Liquid chromatographic chiral separations of the N-6-(endo-2-norbornyl)-9-methyladenine enantiomers. Journal of Chromatography A

[2]. Glover DK, et al. Effect of N-0861, a selective adenosine A1 receptor antagonist, on pharmacologic stress imaging with adenosine. J Nucl Med. 1995 Feb;36(2):270-5.


[Related Small Molecules]

CGS 21680 hydrochloride | Preladenant | ZM 241385 | CPI-444 | SCH 58261 | Vipadenant | Istradefylline | Tozadenant | AZD-4635 | Capadenoson | 2-CL-IB-MECA | PSB-12379 | CD73-IN-1 | IB-MECA | Diprophylline

Chemical & Physical Properties

[ Density]:
1.6±0.1 g/cm3

[ Boiling Point ]:
456.2±48.0 °C at 760 mmHg

[ Molecular Formula ]:
C13H17N5

[ Molecular Weight ]:
243.308

[ Flash Point ]:
229.7±29.6 °C

[ Exact Mass ]:
243.148392

[ LogP ]:
2.17

[ Vapour Pressure ]:
0.0±1.1 mmHg at 25°C

[ Index of Refraction ]:
1.821

[ Storage condition ]:
2-8℃

Related Compounds