PARP1-IN-9
Names
[ CAS No. ]:
2494000-71-2
[ Name ]:
PARP1-IN-9
Biological Activity
[Description]:
PARP1-IN-9 (Compound 5c) is a PARP1 inhibitor with an IC50 of 30.51 nM. PARP1-IN-9 induces cell apoptosis and shows anticancer activity. PARP1-IN-9 has higher potency than Olaparib (HY-10162) [1].
[Related Catalog]:
[Target]
PARP1:30.51 nM (IC50)
[In Vitro]
PARP1-IN-9 (Compound 5c) shows antiproliferative activity with an IC50 of 3.65 μM against MDA-MB-436 cancer cell line[1].
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C18H21N3O5
[ Molecular Weight ]:
359.38