195199-95-2

195199-95-2 structure

Name: SB 258719
Chemical Name: N,3-dimethyl-N-[4-(4-methylpiperidin-1-yl)butan-2-yl]benzenesulfonamide
CAS Number: 195199-95-2
Molecular Formula: C₁₈H₃₀N₂O₂S
Molecular Weight: 338.51
Catalog: Signaling Pathways GPCR/G Protein 5-HT Receptor
Create Date: 2016-04-18 01:48:01
Modify Date: 2024-01-12 17:51:08
SB 258719 is a selective 5-HT7 receptor antagonist with a pKi of 7.5.

Name	N,3-dimethyl-N-[4-(4-methylpiperidin-1-yl)butan-2-yl]benzenesulfonamide
Synonyms	sb-258,719 SB 258719

Description	SB 258719 is a selective 5-HT7 receptor antagonist with a pKi of 7.5.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor Research Areas >> Neurological Disease
Target	pKi: 7.5 (5-HT7 receptor)
References	[1]. Thomas DR, et al. Functional characterisation of the human cloned 5-HT7 receptor (long form); antagonist profile of SB-258719. Br J Pharmacol. 1998 Jul;124(6):1300-6.