1853254-97-3

1853254-97-3 structure
1853254-97-3 structure
  • Name: PEN-221
  • Chemical Name: PEN-221
  • CAS Number: 1853254-97-3
  • Molecular Formula: C83H109ClN14O20S4
  • Molecular Weight: 1786.55
  • Catalog: Signaling Pathways GPCR/G Protein Somatostatin Receptor
  • Create Date: 2019-03-30 19:20:33
  • Modify Date: 2024-01-21 15:57:50
  • PEN-221 is a Somatostatin receptor 2 (SSTR2)-targeting cytotoxic conjugate with an IC50 of 10 nM.

Name PEN-221
Description PEN-221 is a Somatostatin receptor 2 (SSTR2)-targeting cytotoxic conjugate with an IC50 of 10 nM.
Related Catalog
Target

IC50: 10 nM (SSTR2)[1]

References

[1]. White BH, et al. Discovery of an SSTR2-Targeting Maytansinoid Conjugate (PEN-221) with Potent Activity in Vitro and in Vivo. J Med Chem. 2019 Mar 14;62(5):2708-2719.

Molecular Formula C83H109ClN14O20S4
Molecular Weight 1786.55