1416435-96-5

1416435-96-5 structure

Name: GB-88
Chemical Name: GB-88
CAS Number: 1416435-96-5
Molecular Formula: C₃₂H₄₂N₄O₄
Molecular Weight: 546.70
Catalog: Signaling Pathways GPCR/G Protein Protease-Activated Receptor (PAR)
Create Date: 2019-06-05 11:19:34
Modify Date: 2024-01-03 16:15:54
GB-88 is a selective, orally PAR2 antagonist, inhibits PAR2 activates Ca(2+) release with an IC 50 of 2 µM[1].

Name	GB-88

Description	GB-88 is a selective, orally PAR2 antagonist, inhibits PAR2 activates Ca(2+) release with an IC 50 of 2 µM[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Protease-Activated Receptor (PAR) Research Areas >> Inflammation/Immunology
Target	PAR2[1]
References	[1]. Suen JY, et al. Modulating human proteinase activated receptor 2 with a novel antagonist (GB88) and agonist (GB110). Br J Pharmacol. 2012 Mar;165(5):1413-23.