2095160-79-3

2095160-79-3 structure
2095160-79-3 structure
  • Name: SMYD3-IN-1
  • Chemical Name: SMYD3-IN-1
  • CAS Number: 2095160-79-3
  • Molecular Formula: C28H31ClN4O3
  • Molecular Weight: 507.02
  • Catalog: Signaling Pathways Epigenetics Histone Methyltransferase
  • Create Date: 2019-08-04 09:04:58
  • Modify Date: 2024-01-12 16:32:20
  • SMYD3-IN-1 (compound 29) is an irreversible and selective inhibitor of SMYD3 (SET and MYND domain containing 3), with an IC50 of 11.7 nM[1].

Name SMYD3-IN-1
Description SMYD3-IN-1 (compound 29) is an irreversible and selective inhibitor of SMYD3 (SET and MYND domain containing 3), with an IC50 of 11.7 nM[1].
Related Catalog
Target

SMYD3:11.7 nM (IC50)

References

[1]. Huang C, et al. Discovery of Irreversible Inhibitors Targeting Histone Methyltransferase, SMYD3. ACS Med Chem Lett. 2019 May 23;10(6):978-984.

Molecular Formula C28H31ClN4O3
Molecular Weight 507.02