1802226-88-5
1802226-88-5 structure
- Name: PSB-12553
- Chemical Name: PSB-12553
- CAS Number: 1802226-88-5
- Molecular Formula: C18H22N4O9P2S
- Molecular Weight: 532.401
- Create Date: 2020-01-12 11:38:50
- Modify Date: 2024-06-23 15:42:37
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PSB-12553 is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 9.5 nM for rat recombinant eN; displays high selectivity versus other ecto-nucleotidases and ADP-activated P2Y receptors, has high metabolic stability.
| Name | PSB-12553 |
|---|
| Description | PSB-12553 is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 9.5 nM for rat recombinant eN; displays high selectivity versus other ecto-nucleotidases and ADP-activated P2Y receptors, has high metabolic stability. |
|---|---|
| References | References 1. Bhattarai S, et al. J Med Chem. 2015 Aug 13;58(15):6248-63. View Related Products by Target Other Targets |
| Molecular Formula | C18H22N4O9P2S |
|---|---|
| Molecular Weight | 532.401 |