Name | FAUC 1036 |
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Description | A potent, biased allosteric agonist of CXCR3 (pEC50=6.64), selectively induces chemotaxis and receptor internalization, and induces β-arrestin 2 recruitment without any stimulation of G proteins. |
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References | References 1. Milanos L, et al. J Med Chem. 2016 Mar 10;59(5):2222-43. 2. Milanos L, et al. Angew Chem Int Ed Engl. 2016 Dec 5;55(49):15277-15281. View Related Products by Target Chemokine Receptor (CCR and CXCR) |
Molecular Formula | C45H52N4O6 |
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Molecular Weight | 744.933 |