Shanghai Nianxing Industrial Co., Ltd
China
Product Name: PKN1/2-IN-1
Price:
Purity: 98.0%
Stocking Period: 10 Day
Contact: Yang

DC Chemicals Limited
China
Product Name: PKN1/2-IN-1
Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/1g
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

942425-34-5

942425-34-5 structure

942425-34-5 structure

Name: PKN1/2-IN-1
Chemical Name: PKN1/2-IN-1
CAS Number: 942425-34-5
Molecular Formula: C₁₄H₁₅N₃O
Molecular Weight: 241.29
Create Date: 2022-05-20 10:24:51
Modify Date: 2024-04-05 15:35:25
PKN1/2-IN-1 is a potent, cell penetrant and selective PKN2 (PRK2) inhibitor (IC50=16 nM; Ki=8 nM)[1].

Name	PKN1/2-IN-1

Description	PKN1/2-IN-1 is a potent, cell penetrant and selective PKN2 (PRK2) inhibitor (IC50=16 nM; Ki=8 nM)[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Others >> Others
Target	IC50: 16 nM, Ki: 8 nM (PKN2)[1] IC50: 108 nM, Ki: 210 nM (PKN1)[1].
References	[1]. Scott F, et al. Development of dihydropyrrolopyridinone-based PKN2/PRK2 chemical tools to enable drug discovery. Bioorg Med Chem Lett. 2022;60:128588.

Molecular Formula	C₁₄H₁₅N₃O
Molecular Weight	241.29