302952-43-8

302952-43-8 structure
302952-43-8 structure
  • Name: MRGPRX1 agonist 2
  • Chemical Name: MRGPRX1 agonist 2
  • CAS Number: 302952-43-8
  • Molecular Formula: C15H14N2OS
  • Molecular Weight: 270.35
  • Catalog: Research Areas Neurological Disease
  • Create Date: 2022-07-06 18:05:26
  • Modify Date: 2024-01-11 08:43:33
  • MRGPRX1 agonist 2 (compound 1a) is a potent Mas-related G protein-coupled receptor X1 (MRGPRX1) positive allosteric modulator with an EC50 value of 0.48 μM. MRGPRX1 agonist 2 can be used for researching neuropathic pain[1].

Name MRGPRX1 agonist 2
Description MRGPRX1 agonist 2 (compound 1a) is a potent Mas-related G protein-coupled receptor X1 (MRGPRX1) positive allosteric modulator with an EC50 value of 0.48 μM. MRGPRX1 agonist 2 can be used for researching neuropathic pain[1].
Related Catalog
Target

EC50: 0.48 μM (MRGPRX1)[1]

References

[1]. Berhane I, et al. Thieno[2,3-d]pyrimidine-Based Positive Allosteric Modulators of Human Mas-Related G Protein-Coupled Receptor X1 (MRGPRX1). J Med Chem. 2022;65(4):3218-3228.

Molecular Formula C15H14N2OS
Molecular Weight 270.35