2235358-73-1
2235358-73-1 structure
- Name: Deltasonamide 1 TFA
- Chemical Name: Deltasonamide 1 TFA
- CAS Number: 2235358-73-1
- Molecular Formula: C32H40ClF3N6O6S2
- Molecular Weight: 761.27
- Catalog: Signaling Pathways Metabolic Enzyme/Protease Phosphodiesterase (PDE)
- Create Date: 2023-01-17 14:21:26
- Modify Date: 2024-04-02 19:40:13
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Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a KD of 203 pM. Deltasonamide 1 can be used for the research of tumors[1].
| Name | Deltasonamide 1 TFA |
|---|
| Description | Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a KD of 203 pM. Deltasonamide 1 can be used for the research of tumors[1]. |
|---|---|
| Related Catalog | |
| Target |
KD: 203 pM (PDE6δ-KRas)[1] |
| In Vitro | Deltasonamide 1 可以抑制 PDE6δ-KRas，KD 为 203 pM[1]。 Deltasonamide 1 通过多达 7 个氢键与 PDE6δ 结合，产生皮摩尔亲和力[1]。 Deltasonamide 1 强烈减少增殖[1]。 Cell Proliferation Assay[1] Cell Line: RTCA of hPDAC cell lines Concentration: 0.375, 0.75, 1.5, 3, 6, 12 μM Incubation Time: 60 h Result: Inhibited proliferation of human pancreatic cancer cell lines. |
| References |
| Molecular Formula | C32H40ClF3N6O6S2 |
|---|---|
| Molecular Weight | 761.27 |