Name | cetrorelix acetate |
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Description | Cetrorelix Acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM. Sequence: N-acetyl-{2-Naph-Ala}-{Cl-Phe}-{3Py-Ala}-Ser-Tyr-{Cit}-Leu-Arg-Pro-Ala-NH2. |
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Related Catalog | |
Target |
IC50: 1.21 nM GnRH[1]. |
In Vitro | Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells[2]. |
References |
Molecular Formula | C72H96ClN17O16 |
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Molecular Weight | 1491.09000 |
Exact Mass | 1489.69000 |
PSA | 532.97000 |
LogP | 6.02320 |
Storage condition | -20°C |