Name | (4R)-2-Undecyl-4-thiazolidinecarboxylic acid |
---|---|
Synonyms |
2-Undecylthiazolidine-4(R)-carboxylic acid
4-Thiazolidinecarboxylic acid, 2-undecyl-, (4R)- (4R)-2-Undecyl-1,3-thiazolidine-4-carboxylic acid |
Description | CAY10444 (BML-241) is a sphingosine-1-phosphate 3 (S1P3) antagonist. CAY10444 inhibits by 37% S1P-induced increases in Ca2+ in HeLa cells expressing S1P3 receptors[1]. |
---|---|
Related Catalog | |
Target |
S1PR3 |
In Vitro | BML-241 inhibits increases in intracellular Ca2+ concentration via P2 receptor or α1A-adrenoceptor stimulation and α1A-adrenoceptor-mediated contraction of rat mesenteric artery, while it does not affect S1P3-mediated decrease of Forskolin-induced cyclic AMP accumulation[1]. |
References |
Density | 1.0±0.1 g/cm3 |
---|---|
Boiling Point | 439.2±40.0 °C at 760 mmHg |
Molecular Formula | C15H29NO2S |
Molecular Weight | 287.461 |
Flash Point | 219.4±27.3 °C |
Exact Mass | 287.191895 |
PSA | 74.63000 |
LogP | 5.42 |
Vapour Pressure | 0.0±2.3 mmHg at 25°C |
Index of Refraction | 1.495 |
Storage condition | -20°C |
RIDADR | NONH for all modes of transport |
---|---|
HS Code | 2934999090 |
HS Code | 2934999090 |
---|---|
Summary | 2934999090. other heterocyclic compounds. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0% |