Name | 2-methyl-1-(3-morpholin-4-ylpropyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide |
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Synonyms | HC-067047 |
Description | HC-067047 is a potent and selective TRPV4 antagonist with IC50s of 48 nM, 133 nM, and 17 nM for human, rat, and mouse TRPV4. |
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Related Catalog | |
Target |
IC50: 48 nM (human TRPV4), 133 nM (rat TRPV4), 17 nM (mouse TRPV4)[1] |
References |
Molecular Formula | C26H28F3N3O2 |
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Molecular Weight | 471.51500 |
Exact Mass | 471.21300 |
PSA | 49.99000 |
LogP | 5.77880 |
Storage condition | 2-8℃ |
Symbol |
GHS06 |
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Signal Word | Danger |
Hazard Statements | H301-H319 |
Precautionary Statements | P301 + P310-P305 + P351 + P338 |
RIDADR | UN 2811 6.1 / PGIII |