GPR4 antagonist 1

Modify Date: 2024-01-09 10:03:22

GPR4 antagonist 1 Structure
GPR4 antagonist 1 structure
Common Name GPR4 antagonist 1
CAS Number 1197879-16-5 Molecular Weight 431.61600
Density N/A Boiling Point N/A
Molecular Formula C27H37N5 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of GPR4 antagonist 1


GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.

 Names

Name 2-ethyl-3-{4-[(E)-3-(4-isopropylpiperazin-1-yl)prop-1-enyl]benzyl}-5,7-dimethyl-3H-imidazo[4,5-b]pyridine
Synonym More Synonyms

 GPR4 antagonist 1 Biological Activity

Description GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.
Related Catalog
Target

IC50: 189 nM (GPR4)[1].

References

[1]. ARYL SULFONOHYDRAZIDES. US 20090291942 A1.

 Chemical & Physical Properties

Molecular Formula C27H37N5
Molecular Weight 431.61600
Exact Mass 431.30500
PSA 37.19000
LogP 4.57380

 Synonyms

2-Ethyl-3-{4-[(E)-3-(4-isopropyl-piperazin-1-yl)-propenyl]-benzyl}-5,7-dimethyl-3H-imidazo[4,5-b]pyridine
GPR4 RECEPTOR MODULATOR 46