[D-Ala2] -Deltorphin II structure
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Common Name | [D-Ala2] -Deltorphin II | ||
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CAS Number | 122752-16-3 | Molecular Weight | 782.88300 | |
Density | 1.272 g/cm3 | Boiling Point | 1256.2ºC at 760 mmHg | |
Molecular Formula | C38H54N8O10 | Melting Point | N/A | |
MSDS | Chinese USA | Flash Point | 713.5ºC |
Use of [D-Ala2] -Deltorphin IIDeltorphin 2 is a selective peptide agonit for the δ opioid receptor. |
Name | [D-Ala2]-Deltorphin II |
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Synonym | More Synonyms |
Description | Deltorphin 2 is a selective peptide agonit for the δ opioid receptor. |
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Related Catalog | |
Target |
δ opioid receptor[1] |
In Vitro | Deltorphin 2 ([D-Ala2]-Deltorphin II) is enzymatically stable, amphibian heptapeptides that has a high affinity and selectivity for delta-opioid receptor. Deltorphin 2 is the most selective natural delta opioid receptor agonist[1]. |
References |
Density | 1.272 g/cm3 |
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Boiling Point | 1256.2ºC at 760 mmHg |
Molecular Formula | C38H54N8O10 |
Molecular Weight | 782.88300 |
Flash Point | 713.5ºC |
Exact Mass | 782.39600 |
PSA | 301.24000 |
LogP | 2.47290 |
Vapour Pressure | 0mmHg at 25°C |
Index of Refraction | 1.575 |
Storage condition | -20°C |
Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
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RIDADR | NONH for all modes of transport |
Membrane partitioning of various delta-opioid receptor forms before and after agonist activations: the effect of cholesterol.
Biochim. Biophys. Acta 1778(6) , 1483-92, (2008) Lipid rafts depicted as densely packed and thicker membrane microdomains, based on the dynamic clustering of cholesterol and sphingolipids, may help as platforms involved in a wide variety of cellular... |
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Delta opioid receptor-mediated analgesia is not altered in preprotachykinin A knockout mice.
Eur. J. Neurosci. 32(11) , 1921-9, (2010) We have shown that delta opioid receptor (DOPR)-mediated analgesia was enhanced in the complete Freund's adjuvant (CFA) model of inflammation. This effect is thought to originate from translocation of... |
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Functional identification of a novel transport system for endogenous and synthetic opioid peptides in the rabbit conjunctival epithelial cell line CJVE.
Pharm. Res. 26(5) , 1226-35, (2009) To investigate whether conjunctival epithelial cells express transport processes for opioid peptides.We monitored the uptake of [(3)H]deltorphin II and [(3)H]DADLE, two hydrolysis-resistant synthetic ... |
Tyr-D-Ala-Phe-Glu-Val-Val-Gly amide |
M.W. 782.89 C38H54N8O10 |
DELTORPHIN B |
DADELT II |
H-Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2 |
H2N-Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2 |
deltorphin II |
TYR-D-ALA-PHE-GLU-VAL-VAL-GLY-NH2 |
DELTORPHIN II |
Deltorphin 2 |