EP3 antagonist 3

Modify Date: 2024-01-23 15:02:16

EP3 antagonist 3 Structure
EP3 antagonist 3 structure
Common Name EP3 antagonist 3
CAS Number 1227827-88-4 Molecular Weight 362.38
Density N/A Boiling Point N/A
Molecular Formula C21H18N2O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of EP3 antagonist 3


EP3 antagonist 3 (compound 2) is an orally active, potent and selective EP3 antagonist, with a pKi of 8.3. EP3 antagonist 3 shows excellent pharmacokinetic properties. EP3 antagonist 3 can be used for overactive bladder (OAB) research[1].

 Names

Name EP3 antagonist 3

 EP3 antagonist 3 Biological Activity

Description EP3 antagonist 3 (compound 2) is an orally active, potent and selective EP3 antagonist, with a pKi of 8.3. EP3 antagonist 3 shows excellent pharmacokinetic properties. EP3 antagonist 3 can be used for overactive bladder (OAB) research[1].
Related Catalog
Target

EP3 Receptor:8.3 (pKi)

References

[1]. Jin J, et al. Novel 3-Oxazolidinedione-6-aryl-pyridinones as Potent, Selective, and Orally Active EP3 Receptor Antagonists. ACS Med Chem Lett. 2010 May 14;1(7):316-20.

 Chemical & Physical Properties

Molecular Formula C21H18N2O4
Molecular Weight 362.38