CB2R-IN-1

Modify Date: 2024-01-08 18:23:37

CB2R-IN-1 Structure
CB2R-IN-1 structure
Common Name CB2R-IN-1
CAS Number 1257555-79-5 Molecular Weight 608.67
Density N/A Boiling Point N/A
Molecular Formula C23H27F3N4O6S3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CB2R-IN-1


CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.

 Names

Name CB2R-IN-1

 CB2R-IN-1 Biological Activity

Description CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
Related Catalog
Target

CB2 Receptor:0.9 nM (Ki)

In Vitro CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].
References

[1]. Tong L, et al. Expansion of SAR studies on triaryl bis sulfone cannabinoid CB2 receptor ligands. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6785-9.

 Chemical & Physical Properties

Molecular Formula C23H27F3N4O6S3
Molecular Weight 608.67
Storage condition 2-8℃