1257555-79-5

1257555-79-5 structure
1257555-79-5 structure
  • Name: CB2R-IN-1
  • Chemical Name: CB2R-IN-1
  • CAS Number: 1257555-79-5
  • Molecular Formula: C23H27F3N4O6S3
  • Molecular Weight: 608.67
  • Catalog: Signaling Pathways GPCR/G Protein Cannabinoid Receptor
  • Create Date: 2018-01-12 21:37:38
  • Modify Date: 2024-01-08 18:23:37
  • CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.

Name CB2R-IN-1
Description CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
Related Catalog
Target

CB2 Receptor:0.9 nM (Ki)

In Vitro CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].
References

[1]. Tong L, et al. Expansion of SAR studies on triaryl bis sulfone cannabinoid CB2 receptor ligands. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6785-9.

Molecular Formula C23H27F3N4O6S3
Molecular Weight 608.67
Storage condition 2-8℃