Teneligliptin D8

Modify Date: 2024-01-11 11:45:35

Teneligliptin D8 Structure
Teneligliptin D8 structure
Common Name Teneligliptin D8
CAS Number 1391012-95-5 Molecular Weight 434.628
Density 1.4±0.1 g/cm3 Boiling Point 663.4±55.0 °C at 760 mmHg
Molecular Formula C22H22D8N6OS Melting Point N/A
MSDS N/A Flash Point 355.0±31.5 °C

 Use of Teneligliptin D8


Teneligliptin D8 (MP-513 D8) a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting DPP-4 inhibitor[1].

 Names

Name {(2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)(2H8)-1-piperazinyl]-2-pyrrolidinyl}(1,3-thiazolidin-3-yl)methanone
Synonym More Synonyms

 Teneligliptin D8 Biological Activity

Description Teneligliptin D8 (MP-513 D8) a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting DPP-4 inhibitor[1].
Related Catalog
References

[1]. Fukuda-Tsuru S, et al. A novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor, teneligliptin, improves postprandial hyperglycemia and dyslipidemia after single and repeated administrations. Eur J Pharmacol. 2012 Dec 5;696(1-3):194-202.

 Chemical & Physical Properties

Density 1.4±0.1 g/cm3
Boiling Point 663.4±55.0 °C at 760 mmHg
Molecular Formula C22H22D8N6OS
Molecular Weight 434.628
Flash Point 355.0±31.5 °C
Exact Mass 434.270386
LogP 1.15
Vapour Pressure 0.0±2.0 mmHg at 25°C
Index of Refraction 1.721

 Synonyms

Methanone, [(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-1-piperazinyl-2,2,3,3,5,5,6,6-d8]-2-pyrrolidinyl]-3-thiazolidinyl-
{(2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)(2H8)-1-piperazinyl]-2-pyrrolidinyl}(1,3-thiazolidin-3-yl)methanone