AZ 3451
Modify Date: 2024-09-06 11:18:25
AZ 3451 structure
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Common Name | AZ 3451 | ||
|---|---|---|---|---|
| CAS Number | 2100284-59-9 | Molecular Weight | 571.46 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C30H27BrN4O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of AZ 3451AZ3451 is a protease-activated receptor-2 (PAR2) antagonist. |
| Name | AZ3451 |
|---|
| Description | AZ3451 is a protease-activated receptor-2 (PAR2) antagonist. |
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| Related Catalog | |
| Target |
Protease-activated receptor-2[1] |
| In Vitro | Antagonist AZ3451 binds to a remote allosteric site outside the helical bundle of the protease-activated receptor 2. AZ3451 is highly lipophilic, which coincides with the hydrophobic nature of the binding pocket within the membrane. Antagonist binding prevents structural rearrangements required for receptor activation and signalling[1]. |
| References |
| Molecular Formula | C30H27BrN4O3 |
|---|---|
| Molecular Weight | 571.46 |
| Storage condition | 2-8℃ |