LSD1-IN-11p structure
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Common Name | LSD1-IN-11p | ||
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CAS Number | 2101951-67-9 | Molecular Weight | 420.473 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C22H24N6O3 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of LSD1-IN-11pLSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%). |
Name | LSD1-IN-11p |
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Description | LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%). |
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References | References 1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195. View Related Products by Target Histone Demethylase |
Molecular Formula | C22H24N6O3 |
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Molecular Weight | 420.473 |