2035912-43-5

2035912-43-5 structure
2035912-43-5 structure
  • Name: LSD1-IN-6
  • Chemical Name: LSD1-IN-6
  • CAS Number: 2035912-43-5
  • Molecular Formula: C15H13BrN2O3
  • Molecular Weight: 349.18
  • Catalog: Signaling Pathways Epigenetics Histone Demethylase
  • Create Date: 2019-08-03 21:44:59
  • Modify Date: 2024-01-05 16:55:23
  • LSD1-IN-6 (Compound 4m) is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 123 nM. LSD1-IN-6 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1[1].

Name LSD1-IN-6
Description LSD1-IN-6 (Compound 4m) is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 123 nM. LSD1-IN-6 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1[1].
Related Catalog
Target

IC50: 123 nM (LSD1)[1]

References

[1]. Duan YC, et al. Discovery of resveratrol derivatives as novel LSD1 inhibitors: Design, synthesis and their biological evaluation. Eur J Med Chem. 2017 Jan 27;126:246-258.

Molecular Formula C15H13BrN2O3
Molecular Weight 349.18