EHMT2-IN-2

Modify Date: 2024-01-11 10:32:29

EHMT2-IN-2 Structure
EHMT2-IN-2 structure
Common Name EHMT2-IN-2
CAS Number 2230850-47-0 Molecular Weight 374.44
Density N/A Boiling Point N/A
Molecular Formula C21H22N6O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of EHMT2-IN-2


EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer[1].

 Names

Name EHMT2-IN-2

 EHMT2-IN-2 Biological Activity

Description EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer[1].
Related Catalog
Target

EHMTI PEP:<100 nM (IC50)

EHMT2 PEP:<100 nM (IC50)

EHMT2 ICW:<100 nM (IC50)

In Vitro EHMT2-IN-2 (Compound 200) is a potent EHMT inhibitor, with IC50s of all < 100 nM for EEHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].
References

[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1.

 Chemical & Physical Properties

Molecular Formula C21H22N6O
Molecular Weight 374.44
Storage condition 2-8℃