P2Y2R/GPR17 antagonist 1

Modify Date: 2024-01-11 18:31:57

P2Y2R/GPR17 antagonist 1 structure	Common Name	P2Y2R/GPR17 antagonist 1
	CAS Number	2395016-49-4	Molecular Weight	432.83
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₉H₁₃ClN₂O₆S	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of P2Y2R/GPR17 antagonist 1

P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1].

Name	P2Y2R/GPR17 antagonist 1

Description	P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> P2Y Receptor Research Areas >> Inflammation/Immunology
Target	IC50: 1.67 µM (GPR17), 3.17 µM (P2Y2R)[1]
References	[1]. Pillaiyar T, et al. Design, synthesis and biological evaluation of suramin-derived dual antagonists of the proinflammatory G protein-coupled receptors P2Y2 and GPR17. Eur J Med Chem. 2020 Jan 15;186:111789.

Molecular Formula	C₁₉H₁₃ClN₂O₆S
Molecular Weight	432.83

Shanghai Nianxing Industrial Co., Ltd
China
Product Name: P2Y2R/GPR17 antagonist 1
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P2Y2R/GPR17 antagonist 1

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