Name | P2Y2R/GPR17 antagonist 1 |
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Description | P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1]. |
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Related Catalog | |
Target |
IC50: 1.67 µM (GPR17), 3.17 µM (P2Y2R)[1] |
References |
Molecular Formula | C19H13ClN2O6S |
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Molecular Weight | 432.83 |