Tabimorelin hemifumarate

Modify Date: 2024-02-25 13:45:42

Tabimorelin hemifumarate Structure
Tabimorelin hemifumarate structure
Common Name Tabimorelin hemifumarate
CAS Number 242143-80-2 Molecular Weight 586.72
Density N/A Boiling Point N/A
Molecular Formula C32H40N4O3.1/2C4H4O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Tabimorelin hemifumarate


Tabimorelin (NN703) hemifumarate is an orally active growth hormone (GH) secretagogue. Tabimorelin hemifumarate is also a potent inhibitor of CYP3A4 activity[1].

 Names

Name Tabimorelin hemifumarate
Synonym More Synonyms

 Tabimorelin hemifumarate Biological Activity

Description Tabimorelin (NN703) hemifumarate is an orally active growth hormone (GH) secretagogue. Tabimorelin hemifumarate is also a potent inhibitor of CYP3A4 activity[1].
Related Catalog
Target

CYP3A4

References

[1]. Zdravkovic M, et al. A clinical study investigating the pharmacokinetic interaction between NN703 (tabimorelin), a potential inhibitor of CYP3A4 activity, and midazolam, a CYP3A4 substrate. Eur J Clin Pharmacol. 2003 Feb;58(10):683-8.  

 Chemical & Physical Properties

Molecular Formula C32H40N4O3.1/2C4H4O4
Molecular Weight 586.72
Exact Mass 1172.630981

 Synonyms

D-Phenylalaninamide, N-[(2E)-5-amino-5-methyl-1-oxo-2-hexen-1-yl]-N-methyl-3-(2-naphthalenyl)-D-alanyl-N,Nα-dimethyl-, (2E)-2-butenedioate (2:1)
N-[(2E)-5-Amino-5-methyl-2-hexenoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamide (2E)-2-butenedioate (2:1)
Tabimorelin
N-[(2E)-5-Amino-5-methylhex-2-enoyl]-N-methyl-3-(2-naphthyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamide (2E)-but-2-enedioate (2:1)