MRGPRX4 modulator-1

Modify Date: 2024-01-06 10:02:11

MRGPRX4 modulator-1 Structure
MRGPRX4 modulator-1 structure
Common Name MRGPRX4 modulator-1
CAS Number 2492596-61-7 Molecular Weight 359.73
Density N/A Boiling Point N/A
Molecular Formula C16H13ClF3NO3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of MRGPRX4 modulator-1


MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 < 100 nM for MRGPR4. MRGPRX4 modulator-1 can be used for researching MRGPR X4 dependent diseases such as itch, pain, and autoimmune disorders[1].

 Names

Name MRGPRX4 modulator-1

 MRGPRX4 modulator-1 Biological Activity

Description MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 < 100 nM for MRGPR4. MRGPRX4 modulator-1 can be used for researching MRGPR X4 dependent diseases such as itch, pain, and autoimmune disorders[1].
Related Catalog
Target

IC50: < 100 nM (MRGPR X4)[1]

References

[1]. Adam YEAGER, et al. Modulators of mas-related g-protein receptor x4 and related products and methods. WO2020198537 (compound 31-2).

 Chemical & Physical Properties

Molecular Formula C16H13ClF3NO3
Molecular Weight 359.73