2492596-61-7

2492596-61-7 structure
2492596-61-7 structure
  • Name: MRGPRX4 modulator-1
  • Chemical Name: MRGPRX4 modulator-1
  • CAS Number: 2492596-61-7
  • Molecular Formula: C16H13ClF3NO3
  • Molecular Weight: 359.73
  • Catalog: Research Areas Inflammation/Immunology
  • Create Date: 2022-07-02 19:11:44
  • Modify Date: 2024-01-06 10:02:11
  • MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 < 100 nM for MRGPR4. MRGPRX4 modulator-1 can be used for researching MRGPR X4 dependent diseases such as itch, pain, and autoimmune disorders[1].

Name MRGPRX4 modulator-1
Description MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 < 100 nM for MRGPR4. MRGPRX4 modulator-1 can be used for researching MRGPR X4 dependent diseases such as itch, pain, and autoimmune disorders[1].
Related Catalog
Target

IC50: < 100 nM (MRGPR X4)[1]

References

[1]. Adam YEAGER, et al. Modulators of mas-related g-protein receptor x4 and related products and methods. WO2020198537 (compound 31-2).

Molecular Formula C16H13ClF3NO3
Molecular Weight 359.73