ESI 05 structure
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Common Name | ESI 05 | ||
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CAS Number | 5184-64-5 | Molecular Weight | 274.37800 | |
Density | 1.129g/cm3 | Boiling Point | 426.7ºC at 760mmHg | |
Molecular Formula | C16H18O2S | Melting Point | N/A | |
MSDS | N/A | Flash Point | 250ºC |
Use of ESI 05ESI-05 (NSC 116966) is a specific exchange protein directly activated by cAMP 2 (EPAC2) antagonist (IC50, 0.4 µM), suppresses the cAMP-mediated activation of EPAC2 and inhibits Rap1 activation mediated by EAPC2[1]. |
Name | 1,3,5-trimethyl-2-(4-methylphenyl)sulfonylbenzene |
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Synonym | More Synonyms |
Description | ESI-05 (NSC 116966) is a specific exchange protein directly activated by cAMP 2 (EPAC2) antagonist (IC50, 0.4 µM), suppresses the cAMP-mediated activation of EPAC2 and inhibits Rap1 activation mediated by EAPC2[1]. |
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Related Catalog | |
Target |
IC50: 0.4 µM (EPAC2)[1] |
References |
Density | 1.129g/cm3 |
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Boiling Point | 426.7ºC at 760mmHg |
Molecular Formula | C16H18O2S |
Molecular Weight | 274.37800 |
Flash Point | 250ºC |
Exact Mass | 274.10300 |
PSA | 42.52000 |
LogP | 4.83380 |
Index of Refraction | 1.562 |
Precursor 10 | |
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DownStream 0 |
mesityl(4-methylphenyl) sulfone |