OMDM-5

Modify Date: 2024-01-30 18:10:09

OMDM-5 Structure
OMDM-5 structure
Common Name OMDM-5
CAS Number 616884-66-3 Molecular Weight 432.64
Density N/A Boiling Point N/A
Molecular Formula C26H44N2O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of OMDM-5


OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1].

 Names

Name OMDM-5

 OMDM-5 Biological Activity

Description OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1].
Related Catalog
Target

Ki: 4.8 μM (anandamide cellular uptake), 4.9 μM (CB1), EC50: 75 nM (VR1)[1]

References

[1]. Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65(9):1473-81.

 Chemical & Physical Properties

Molecular Formula C26H44N2O3
Molecular Weight 432.64
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