OMDM-5 structure
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Common Name | OMDM-5 | ||
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CAS Number | 616884-66-3 | Molecular Weight | 432.64 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C26H44N2O3 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of OMDM-5OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1]. |
Name | OMDM-5 |
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Description | OMDM-5 is a selective inhibitor of anandamide cellular uptake (ACU), with a Ki of 4.8 μM. OMDM-5 is also a potent vanilloid receptor type 1 (VR1, TRPV1) agonist, with an EC50 of 75 nM, and shows weakly active as cannabinoid receptor type 1 (CB1) ligand (Ki=4.9 μM)[1]. |
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Related Catalog | |
Target |
Ki: 4.8 μM (anandamide cellular uptake), 4.9 μM (CB1), EC50: 75 nM (VR1)[1] |
References |
Molecular Formula | C26H44N2O3 |
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Molecular Weight | 432.64 |