[D- MET2 , PRO5 ]-ENKEPHALINAMIDE structure
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Common Name | [D- MET2 , PRO5 ]-ENKEPHALINAMIDE | ||
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CAS Number | 63307-63-1 | Molecular Weight | 612.74000 | |
Density | 1.31g/cm3 | Boiling Point | 1065ºC at 760 mmHg | |
Molecular Formula | C30H40N6O6S | Melting Point | N/A | |
MSDS | N/A | Flash Point | 597.9ºC |
Use of [D- MET2 , PRO5 ]-ENKEPHALINAMIDE(D-Met2,Pro5)-Enkephalinamide is a highly potent opiate agonist, and shows antinociceptive activity[1][2][3]. |
Name | 1-[2-[[2-[[2-[[2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylsulfanylbutanoyl]amino]acetyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxamide |
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Synonym | More Synonyms |
Description | (D-Met2,Pro5)-Enkephalinamide is a highly potent opiate agonist, and shows antinociceptive activity[1][2][3]. |
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Related Catalog | |
In Vivo | (D-Met2,Pro5)-Enkephalinamide (intravenous injection; 0.25 and 0.5 mg/kg; once) leads to the decreasement of prolactin (PRL) secretion in lactating rats[2]. Animal Model: Wistar lactating rats[2] Dosage: 0.25 and 0.5 mg/kg Administration: Intravenous injection; 0.25 and 0.5 mg/kg; once Result: Decreased plasma PRL levels 15 min after the administration in continuously lactating rats. Produced a marked depression in plasma PRL concentration in non-deprived lactating mothers. |
Density | 1.31g/cm3 |
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Boiling Point | 1065ºC at 760 mmHg |
Molecular Formula | C30H40N6O6S |
Molecular Weight | 612.74000 |
Flash Point | 597.9ºC |
Exact Mass | 612.27300 |
PSA | 233.71000 |
LogP | 4.12870 |
Index of Refraction | 1.616 |
CHEMICAL IDENTIFICATION
HEALTH HAZARD DATAACUTE TOXICITY DATA
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~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
~% [D- MET2 , PRO5... CAS#:63307-63-1 |
Literature: Audigier; Mazarguil; Gout; Cros European Journal of Medicinal Chemistry, 1980 , vol. 15, # 2 p. 173 - 177 |
H-Tyr-D-Met-Gly-Phe-Pro-NH2 |
L-tyrosyl-D-methionyl-glycyl-L-phenylalanyl-L-proline amide |
Tyr-D-Met-Gly-Phe-Pro-NH2 |