Didesmethyl cariprazine

Modify Date: 2024-01-06 10:25:05

Didesmethyl cariprazine Structure
Didesmethyl cariprazine structure
Common Name Didesmethyl cariprazine
CAS Number 839712-25-3 Molecular Weight 399.36
Density N/A Boiling Point N/A
Molecular Formula C19H28Cl2N4O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Didesmethyl cariprazine


Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic drug candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor[1].

 Names

Name Didesmethyl cariprazine

 Didesmethyl cariprazine Biological Activity

Description Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic drug candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor[1].
Related Catalog
References

[1]. Citrome L, et al. Cariprazine for acute and maintenance treatment of adults with schizophrenia: an evidence-based review and place in therapy. Neuropsychiatr Dis Treat. 2018 Oct 5;14:2563-2577.

 Chemical & Physical Properties

Molecular Formula C19H28Cl2N4O
Molecular Weight 399.36