839712-25-3

839712-25-3 structure

Name: Didesmethyl cariprazine
Chemical Name: Didesmethyl cariprazine
CAS Number: 839712-25-3
Molecular Formula: C₁₉H₂₈Cl₂N₄O
Molecular Weight: 399.36
Catalog: Signaling Pathways GPCR/G Protein 5-HT Receptor
Create Date: 2020-01-23 17:43:51
Modify Date: 2024-01-06 10:25:05
Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic drug candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor[1].

Name	Didesmethyl cariprazine

Description	Didesmethyl cariprazine is a metabolite of Cariprazine and acts as the predominant circulating active moiety. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a antipsychotic drug candidate that exhibits high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Dopamine Receptor Signaling Pathways >> Neuronal Signaling >> Dopamine Receptor Research Areas >> Neurological Disease Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor
References	[1]. Citrome L, et al. Cariprazine for acute and maintenance treatment of adults with schizophrenia: an evidence-based review and place in therapy. Neuropsychiatr Dis Treat. 2018 Oct 5;14:2563-2577.

Molecular Formula	C₁₉H₂₈Cl₂N₄O
Molecular Weight	399.36