Cyclobenzaprine-d6 hydrochloride

Modify Date: 2024-01-10 09:27:03

Cyclobenzaprine-d6 hydrochloride Structure
Cyclobenzaprine-d6 hydrochloride structure
Common Name Cyclobenzaprine-d6 hydrochloride
CAS Number 2748492-38-6 Molecular Weight 317.89
Density N/A Boiling Point N/A
Molecular Formula C20H16D6ClN Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Cyclobenzaprine-d6 hydrochloride


Cyclobenzaprine-d6 (hydrochloride) is deuterium labeled Cyclobenzaprine (hydrochloride).

 Names

Name Cyclobenzaprine-d6 hydrochloride

 Cyclobenzaprine-d6 hydrochloride Biological Activity

Description Cyclobenzaprine-d6 (hydrochloride) is deuterium labeled Cyclobenzaprine (hydrochloride).
Related Catalog
In Vitro Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216.

[2]. Kobayashi, H., Y. Hasegawa, and H. Ono, Cyclobenzaprine, a centrally acting muscle relaxant, acts on descending serotonergic systems. Eur J Pharmacol, 1996. 311(1): p. 29-35.

[3]. Honda, M., T. Nishida, and H. Ono, Tricyclic analogs cyclobenzaprine, amitriptyline and cyproheptadine inhibit the spinal reflex transmission through 5-HT(2) receptors. Eur J Pharmacol, 2003. 458(1-2): p. 91-9.

 Chemical & Physical Properties

Molecular Formula C20H16D6ClN
Molecular Weight 317.89