GSK215083

Modify Date: 2024-01-10 04:50:12

GSK215083 Structure
GSK215083 structure
Common Name GSK215083
CAS Number 607742-80-3 Molecular Weight 385.46
Density N/A Boiling Point N/A
Molecular Formula C20H20FN3O2S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of GSK215083


GSK215083 is a high affinity 5-HT6 receptor antagonist. GSK215083 can serves as a promising 5-HT6 radioligand candidate by radiolabeled with (11)C via methylation[1].

 Names

Name 4-(3-fluorophenyl)sulfonyl-8-(4-methylpiperazin-1-yl)quinoline
Synonym More Synonyms

 GSK215083 Biological Activity

Description GSK215083 is a high affinity 5-HT6 receptor antagonist. GSK215083 can serves as a promising 5-HT6 radioligand candidate by radiolabeled with (11)C via methylation[1].
Related Catalog
Target

5-HT6 Receptor

References

[1]. Parker CA, et al. Radiosynthesis and characterization of 11C-GSK215083 as a PET radioligand for the 5-HT6 receptor. J Nucl Med. 2012 Feb;53(2):295-303.  

 Chemical & Physical Properties

Molecular Formula C20H20FN3O2S
Molecular Weight 385.46
Exact Mass 385.12600
PSA 61.89000
LogP 4.04220

 Synonyms

unii-8gfe8j4n0z