Blue FPG-A trisodium

Modify Date: 2024-09-17 21:18:07

Blue FPG-A trisodium Structure
Blue FPG-A trisodium structure
Common Name Blue FPG-A trisodium
CAS Number 78617-94-4 Molecular Weight 840.10
Density N/A Boiling Point N/A
Molecular Formula C29H17ClN7Na3O11S3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Blue FPG-A trisodium


Blue FPG-A trisodium is a selective antagonist of P2X1 receptor and P2Y1 receptor with IC50 values of 35.5 μM and 2.6 μM, respectively. Blue FPG-A trisodium is a structural isomer of the components of Reactive Blue 2 (RB2)[1].

 Names

Name Blue FPG-A trisodium

 Blue FPG-A trisodium Biological Activity

Description Blue FPG-A trisodium is a selective antagonist of P2X1 receptor and P2Y1 receptor with IC50 values of 35.5 μM and 2.6 μM, respectively. Blue FPG-A trisodium is a structural isomer of the components of Reactive Blue 2 (RB2)[1].
Related Catalog
Target

p2x1 Receptor:35.5 μM (IC50)

P2Y1 Receptor:2.6 μM (IC50)

In Vitro Blue FPG-A trisodium (RB 2 para) (1、3.2、10、32 和 100 μM) 抑制 α、β-亚甲基 ATP (α、β-MeATP) 诱导的大鼠输精管 (RVD) 收缩和 5’-o-(2-硫代二磷酸腺苷) (ADPβS) 诱导的卡巴胆碱 (Carbachol,HY-B1208) 预处理的豚鼠大肠带绦虫 (GPTC) 的松弛[1]。
References

[1]. Glänzel M, et al. Constitutional isomers of Reactive Blue 2 - selective P2Y-receptor antagonists? Eur J Med Chem. 2003 Mar;38(3):303-12.  

 Chemical & Physical Properties

Molecular Formula C29H17ClN7Na3O11S3
Molecular Weight 840.10