Farampator-d10

Modify Date: 2024-01-14 08:34:27

Farampator-d10 Structure
Farampator-d10 structure
Common Name Farampator-d10
CAS Number 211735-93-2 Molecular Weight 241.31
Density N/A Boiling Point N/A
Molecular Formula C12H3D10N3O2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Farampator-d10


Farampator-d10 (CX-691-d10) is the deuterium labeled Farampator. Farampator (CX-691) is an AMPA receptor positive modulator.

 Names

Name Farampator-d10

 Farampator-d10 Biological Activity

Description Farampator-d10 (CX-691-d10) is the deuterium labeled Farampator. Farampator (CX-691) is an AMPA receptor positive modulator.
Related Catalog
In Vitro Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216.

[2]. Woolley ML, et al. Evaluation of the pro-cognitive effects of the AMPA receptor positive modulator, 5-(1-piperidinylcarbonyl)-2,1,3-benzoxadiazole (CX691), in the rat. Psychopharmacology (Berl). 2009 Jan;202(1-3):343-54.

[3]. Wezenberg E, et al. Acute effects of the ampakine farampator on memory and information processing in healthy elderly volunteers. Neuropsychopharmacology. 2007 Jun;32(6):1272-83.

 Chemical & Physical Properties

Molecular Formula C12H3D10N3O2
Molecular Weight 241.31