36840-10-5
36840-10-5 structure
- Name: LPA2 antagonist 2
- Chemical Name: 4,4'-(4,4'-Biphenyldiyldiimino)Bis(4-Oxo-2-Butenoic Acid)
- CAS Number: 36840-10-5
- Molecular Formula: C20H16N2O6
- Molecular Weight: 380.35100
- Catalog: Signaling Pathways GPCR/G Protein LPL Receptor
- Create Date: 2018-02-28 21:30:01
- Modify Date: 2024-01-10 13:23:25
-
LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is ＞480-fold more selective than LPA3 (IC50 of 13.85 μM)[1].
| Name | 4,4'-(4,4'-Biphenyldiyldiimino)Bis(4-Oxo-2-Butenoic Acid) |
|---|---|
| Synonyms | MFCD00566434 |
| Description | LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is ＞480-fold more selective than LPA3 (IC50 of 13.85 μM)[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 28.3 nM (LPA2); 13.85 μM (LPA3)[1] |
| References |
| Density | 1.444±0.06 g/cm3(Predicted) |
|---|---|
| Boiling Point | 758.0±60.0 °C(Predicted) |
| Molecular Formula | C20H16N2O6 |
| Molecular Weight | 380.35100 |
| Exact Mass | 380.10100 |
| PSA | 132.80000 |
| LogP | 2.65820 |
| Storage condition | 2-8°C |