866206-55-5
866206-55-5 structure
- Name: PRX-08066 Maleic acid
- Chemical Name: 5-({4-[(6-Chlorothieno[2,3-d]pyrimidin-4-yl)amino]-1-piperidinyl} methyl)-2-fluorobenzonitrile (2Z)-2-butenedioate (1:1)
- CAS Number: 866206-55-5
- Molecular Formula: C23H21ClFN5O4S
- Molecular Weight: 517.96
- Catalog: Biochemical Inhibitor Neuronal Signaling 5-HT Receptor Antagonist
- Create Date: 2016-12-07 17:19:50
- Modify Date: 2024-01-24 17:47:53
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PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that causes selective vasodilation of pulmonary arteries.
| Name | 5-({4-[(6-Chlorothieno[2,3-d]pyrimidin-4-yl)amino]-1-piperidinyl} methyl)-2-fluorobenzonitrile (2Z)-2-butenedioate (1:1) |
|---|---|
| Synonyms |
Benzonitrile, 5-[[4-[(6-chlorothieno[2,3-d]pyrimidin-4-yl)amino]-1-piperidinyl]methyl]-2-fluoro-, (2Z)-2-butenedioate (1:1)
5-({4-[(6-Chlorothieno[2,3-d]pyrimidin-4-yl)amino]-1-piperidinyl}methyl)-2-fluorobenzonitrile (2Z)-2-butenedioate (1:1) |
| Description | PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that causes selective vasodilation of pulmonary arteries. |
|---|---|
| Related Catalog | |
| Target |
5-HT2B Receptor:3.4 nM (IC50) |
| Molecular Formula | C23H21ClFN5O4S |
|---|---|
| Molecular Weight | 517.96 |
| Exact Mass | 517.098694 |
| PSA | 167.68000 |
| LogP | 4.15468 |
| Storage condition | -20℃ |