1637770-13-8
1637770-13-8 structure
- Name: GS-626510
- Chemical Name: GS-626510
- CAS Number: 1637770-13-8
- Molecular Formula: C25H22N4O
- Molecular Weight: 394.47
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2019-03-30 13:20:33
- Modify Date: 2024-01-10 20:15:11
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GS-626510 is a potent, and orally bioavailable BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively[1].
| Name | GS-626510 |
|---|
| Description | GS-626510 is a potent, and orally bioavailable BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively[1]. |
|---|---|
| Related Catalog | |
| Target |
BRD2:0.59-2.5 nM (Kd) BRD3:0.65-0.66 nM (Kd) BRD4:1.3-3.2 nM (Kd) BD1:83 nM (IC50) BD2:78 nM (IC50) |
| References |
| Molecular Formula | C25H22N4O |
|---|---|
| Molecular Weight | 394.47 |