2180931-09-1
2180931-09-1 structure
- Name: CARM1 inhibitor 9
- Chemical Name: CARM1 inhibitor 9
- CAS Number: 2180931-09-1
- Molecular Formula: C15H24BrN3
- Molecular Weight: 326.282
- Create Date: 2020-01-20 15:57:56
- Modify Date: 2024-01-07 19:39:22
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CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM; displays 20-fold selective for CARM1 over PRMT6 and highly selective over PRMT1, PRMT3, PRMT8 as well as PRMT5 and PRMT7; CARM1 inhibitor 9 is a useful tool for studying the role of CARM1 in health and disease.
| Name | CARM1 inhibitor 9 |
|---|
| Description | CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM; displays 20-fold selective for CARM1 over PRMT6 and highly selective over PRMT1, PRMT3, PRMT8 as well as PRMT5 and PRMT7; CARM1 inhibitor 9 is a useful tool for studying the role of CARM1 in health and disease. |
|---|---|
| References | References 1. Kaniskan HÜ, et al. Medchemcomm. 2016 Sep 1;7(9):1793-1796. View Related Products by Target Histone Methyltransferase (HMTase) |
| Molecular Formula | C15H24BrN3 |
|---|---|
| Molecular Weight | 326.282 |